Kitasamycin Tartrate Soluble Powder
Gitarimisin
Produk iki bubuk putih utawa meh putih.
Pharmacodynamics Guitarimycin kalebu antibiotik macrolide, kanthi spektrum antibakteri sing padha karo eritromisin, lan mekanisme tumindake padha karo eritromisin. Bakteri gram-positif sing sensitif kalebu Staphylococcus aureus (kalebu Staphylococcus aureus sing tahan penisilin), pneumococcus, streptococcus, anthrax, erysipelas suis, listeria, clostridium putrescence, clostridium anthracis, lsp. Kajaba iku, uga duwe efek apik ing mycoplasma. Efek antibakteri tumrap bakteri gram-positif sing umume rada kalah karo bakteri gram-positif.
Erythromycin duweni efek antibakteri sing padha ing mycoplasma karo tylosin, lan uga efektif ing rickettsia lan spirochetes.
Efek saka Staphylococcus aureus sing tahan luwih apik tinimbang erythromycin lan tetracycline. Farmakokinetik diserep kanthi apik sawise administrasi oral lan tekan konsentrasi puncak ing getih sawise 2 jam. Disebarake sacara wiyar ing organ utama, ing antarane konsentrasi ing ati, paru-paru, ginjel lan otot luwih dhuwur tinimbang ing getih. Utamane diekskresi liwat sistem hepatobiliary, kanthi konsentrasi dhuwur ing empedu lan feces. Jumlah cilik diekskresi liwat ginjel.
(1) Amarga saka target padha, iku ngirim ora digunakake bebarengan karo macrolides liyane, amina linco lan alkohol amida.
(2) Yen digabungake karo B-laktam, nduweni efek antagonis.
Antibiotik macrolide. Utamane digunakake kanggo nambani penyakit infèksi sing disebabake dening bakteri gram positif, mycoplasma, lan liya-liyane.
Diwilang dening prodhuk iki. Ngombé campuran: 2,5 ~ 5g pitik saben 1L banyu. Bisa digunakake terus-terusan kanggo 3 ~ 5 dina.
Sawise administrasi lisan, kewan bisa ngalami disfungsi gastrointestinal gumantung dosis (kayata muntah, diare, nyeri usus, lan liya-liyane), kanthi insiden sing luwih murah tinimbang eritromisin.
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