I-Kitasamycin Tartrate Umgubo onyibilikayo
Guitarimycin
Le mveliso imhlophe okanye iphantse ibe ngumgubo omhlophe.
I-Pharmacodynamics Guitarimycin yeye-macrolide antibiotics, ene-antibacterial spectrum efana ne-erythromycin, kwaye indlela yokusebenza iyafana ne-erythromycin. Iintsholongwane zegram-positive zibandakanya i-Staphylococcus aureus (kuquka i-penicillin resistant Staphylococcus aureus), i-pneumococcus, i-streptococcus, i-anthrax, i-erysipelas suis, i-listeria, i-clostridium putrescence, i-clostridium anthracis, njl. I-Sensitive influngococcuses, i-Haephilus influosteococcus, i-influngococcus, i-influngococcus, i-anthracis , njl. Ukongeza, inefuthe elihle kwi-mycoplasma. Impembelelo ye-antibacterial ngokuchasene nebhaktiriya eninzi yegram-positive ingaphantsi kancinane kunebhaktheriya yegram-positive.
I-Erythromycin inefuthe elifanayo le-antibacterial kwi-mycoplasma ukuya kwi-tylosin, kwaye iyasebenza kwi-rickettsia kunye ne-spirochetes.
Impembelelo ye-Staphylococcus aureus enganyangekiyo yayingcono kune-erythromycin kunye ne-tetracycline. I-pharmacokinetics yaxutywa kakuhle emva kokulawulwa komlomo kwaye yafikelela kwi-concentration concentration kwi-2 iiyure kamva. Isasazwa ngokubanzi kwizitho eziphambili, phakathi kwazo ukugxilwa kwesibindi, imiphunga, izintso kunye nezihlunu ziphezulu kunegazi. Ininzi ikhutshwe nge-hepatobiliary system, kunye nokugxininiswa okuphezulu kwi-bile kunye nendle. Isixa esincinci sikhutshwa ngentso.
(1) Ngenxa yenjongo efanayo, akufanele isetyenziswe ngexesha elifanayo njengamanye ama-macrolides, i-linco amines kunye ne-amide alcohols.
(2) Xa idibene ne-B-lactam, inefuthe elichasayo.
Macrolide antibiotics. Ikakhulu isetyenziselwa ukunyanga izifo ezithathelwanayo ezibangelwa iibhaktheriya zegram-positive, i-mycoplasma, njl.
Kubalwa yile mveliso. Ukusela okuxutyiweyo: 2.5 ~ 5g yenkukhu nge-1L yamanzi. Ingasetyenziswa ngokuqhubekayo kwi-3 ~ 5 iintsuku.
Emva kokulawulwa komlomo, izilwanyana zinokuba ne-dose exhomekeke kwi-gastrointestinal dysfunction (njengokuhlanza, isifo sohudo, intlungu yamathumbu, njl.), kunye nesiganeko esisezantsi kune-erythromycin.
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