Amoxicillin soluble ntụ ntụ
Amoxicillin
Ngwaahịa a dị ọcha ma ọ bụ ihe fọrọ nke nta ka ọ bụrụ ntụ ntụ.
Pharmacodynamics Amoxicillin bụ ọgwụ nje B-lactam nwere mmetụta nje bacteria sara mbara. Ụdị dị iche iche nke nje bacteria na ọrụ bụ otu ihe ahụ na ampicillin. Ọrụ antibacterial megide ọtụtụ nje bacteria nwere gram dị ntakịrị ike karịa penicillin, ọ na-enwe mmetụta nke penicillinase, ya mere ọ dịghị arụ ọrụ na penicillin na-eguzogide Staphylococcus aureus. Ọ na-enwe mmetụta siri ike na nje bacteria gram-adịghị mma dị ka Escherichia coli, Proteus, Salmonella, Haemophilus, Brucella na Pasteurella, ma nje bacteria ndị a na-enwekarị mgbochi ọgwụ. Ọ naghị emetụta Pseudomonas aeruginosa. N'ihi na mmịnye ya na anụmanụ monogastric dị mma karịa ampicillin, na ntinye ọbara ya dị elu, ọ na-enwe mmetụta dị mma na ọrịa sistem. Ọ na-emetụta usoro iku ume, usoro urinary, akpụkpọ anụ na anụ ahụ dị nro nke nje bacteria na-emetụ n'ahụ kpatara.
Pharmacokinetics: amoxicillin kwụsiri ike na acid gastric, nke a na-etinye ya na 74% ~ 92% mgbe nchịkwa ọnụ na anụmanụ monogastric. Ihe dị n'ime eriri afọ eriri afọ na-emetụta ọnụ ọgụgụ absorption, ma ọ dịghị emetụta ogo nke absorption, ya mere enwere ike iji nri agwakọta. Mgbe nchịkwa ọnụ nke otu dose gasịrị, ntinye uche nke amoxicillin dị elu ugboro 1.5-3 karịa nke ampicillin.
(1) Nchikota nke ngwaahịa a na aminoglycosides nwere ike ime ka ntinye nke ikpeazụ na nje bacteria na-egosi mmetụta synergistic.
(2) Ngwa ngwa bacteriostatic agents dị ka macrolides, tetracyclines na amide alcohols na-egbochi mmetụta bactericidal nke ngwaahịa a ma ghara ijikọ ọnụ.
β-Lactam ọgwụ nje. A na-eji ya agwọ ọrịa nje bacteria gram-positive na gram-negative bacteria nwere mmetụta nke amoxicillin na ọkụkọ.
Ngwaahịa a gbakọrọ ya. Were ọnụ: 0.2 ~ 0.3g ọkụkọ kwa 1kg arọ ahụ. 2 ugboro n'ụbọchị maka 5 consecutive ụbọchị: agwakọta ihe ọṅụṅụ: 0,6g ọkụkọ kwa 1L mmiri maka 3 ka 5 consecutive ụbọchị.
Ọ nwere mmetụta nnyonye anya siri ike na ahịhịa nkịtị nke eriri afọ.
(1) A gaghị eji ọkụkọ na-akụ akwa maka oriri mmadụ n'oge ịtọgbọ.
(2) E kwesịghị iji gram positive bacteria na-eguzogide penicillin.
(3) Dị njikere iji.
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