ʻO Amoxicillin Soluble Powder
ʻO Amoxicillin
He keʻokeʻo a aneane keʻokeʻo kēia huahana.
ʻO Pharmacodynamics Amoxicillin kahi lāʻau antibiotic B-lactam me ka hopena antibacterial ākea ākea. ʻO ke ʻano o ka antibacterial spectrum a me ka hana like ʻole me ka ampicillin. ʻOi aku ka nāwaliwali o ka hana antibacterial e kūʻē i ka hapa nui o nā huakini gram-positive ma mua o ka penicillin, a ua maʻalahi ia i ka penicillinase, no laila ʻaʻole kūpono ia i ka penicillin resistant Staphylococcus aureus. He hopena koʻikoʻi ma luna o nā hua bacteria gram-negative e like me Escherichia coli, Proteus, Salmonella, Haemophilus, Brucella a me Pasteurella, akā hiki i kēia mau bacteria ke kū'ē i ka lāʻau. ʻAʻole pili ia i ka Pseudomonas aeruginosa. No ka mea, ʻoi aku ka maikaʻi o kona komo ʻana i loko o nā holoholona monogastric ma mua o ka ampicillin, a ʻoi aku ka kiʻekiʻe o ke koko, ʻoi aku ka maikaʻi o ka hopena i ka maʻi ʻōnaehana. Pili ia i ka ʻōnaehana hanu, ka ʻōnaehana urinary, ka ʻili a me nā maʻi ʻiʻo palupalu i hoʻokumu ʻia e ka maʻi bacteria.
Pharmacokinetics: paʻa loa ka amoxicillin i ka waikawa gastric, ka mea i hoʻopili ʻia e 74% ~ 92% ma hope o ka hoʻokele waha i nā holoholona monogastric. Hoʻopili nā mea i loko o ka ʻōpū o ka ʻōpū i ka absorption rate, akā ʻaʻole pili i ke kiʻekiʻe o ka absorption, no laila hiki ke hoʻohana ʻia i ka hānai ʻana. Ma hope o ka hoʻohana waha ʻana i ka nui like, ʻo ka nui o ka serum o ka amoxicillin he 1.5-3 mau manawa kiʻekiʻe ma mua o ka ampicillin.
(1) Hiki i ka hui pū ʻana o kēia huahana a me nā aminoglycosides ke hoʻonui i ka manaʻo o ka hope i loko o ka bacteria, e hōʻike ana i kahi hopena synergistic.
(2) ʻO nā mea hana bacteriostatic wikiwiki e like me nā macrolides, tetracyclines a me nā amide alcohols e hoʻopilikia i ka hopena bactericidal o kēia huahana a ʻaʻole pono e hoʻohana pū ʻia.
β- Lactam nā lāʻau lapaʻau. Hoʻohana ʻia ia e mālama i ka maʻi o ka maʻi bacteria gram-positive a me ka bacteria gram-negative i pili i ka amoxicillin i loko o nā moa.
Ua helu ʻia e kēia huahana. E lawe waha: 0.2~0.3g moa no 1kg kaumaha o ke kino. 2 manawa i ka lā no 5 mau lā: inu hui: 0.6g moa no 1L wai no 3 a 5 mau lā.
Loaʻa iā ia ka hopena interference ikaika i ka flora maʻamau o ka gastrointestinal tract.
(1) ʻAʻole e hoʻohana ʻia nā moa e hoʻomoe ana i nā hua no ka ʻai kanaka i ka wā hoʻomoe.
(2) ʻAʻole pono e hoʻohana ʻia nā hua bacteria Gram positive kūʻē i ka penicillin.
(3) Mākaukau e hoʻohana.
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