I-Amoxicillin Umgubo onyibilikayo
Amoxicillin
Le mveliso imhlophe okanye iphantse ibe ngumgubo omhlophe.
I-Pharmacodynamics I-Amoxicillin yi-antibiotic ye-B-lactam ene-antibacterial effect ebanzi. I-antibacterial spectrum kunye nomsebenzi ngokusisiseko ziyafana ne-ampicillin. Umsebenzi we-antibacterial ngokuchasene neebhaktheriya ezininzi ezinegram ubuthathaka kancinci kune-penicillin, kwaye inovelwano kwi-penicillinase, ngoko ke ayisebenzi kwi-penicillin ekwaziyo ukumelana ne-Staphylococcus aureus. Inempembelelo eyomeleleyo kwiibhaktiriya ezinegram-negative ezifana ne-Escherichia coli, i-Proteus, i-Salmonella, i-Haemophilus, i-Brucella kunye ne-Pasteurella, kodwa ezi bhaktiriya ziyakwazi ukumelana namachiza. Ayinabungozi kwiPseudomonas aeruginosa. Ngenxa yokuba ukufunxwa kwayo kwizilwanyana ze-monogastric kungcono kune-ampicillin, kwaye ukuxinwa kwayo kwegazi kuphezulu, kunempembelelo engcono kusulelo lwenkqubo. Isebenza kwinkqubo yokuphefumla, inkqubo yomchamo, ulusu kunye nosulelo lwezicubu ezithambileyo ezibangelwa ziibhaktheriya ezibuthathaka.
I-Pharmacokinetics: i-amoxicillin izinzile kwi-asidi yesisu, efunxwa yi-74% ~ 92% emva kokulawulwa komlomo kwizilwanyana ze-monogastric. Imixholo yendlela yesisu ichaphazela izinga lokufunxa, kodwa ayichaphazeli iqondo lokufunxa, ngoko ke ukutya okuxutyiweyo kungasetyenziswa. Emva kokulawulwa komlomo kwidosi efanayo, i-serum yoxinaniso ye-amoxicillin yayiyi-1.5 ~ 3 amaxesha aphezulu kune-ampicillin.
(1) Ukudibanisa le mveliso kunye ne-aminoglycosides kunokunyusa ukuxinwa kokugqibela kwiibhaktheriya, kubonisa umphumo we-synergistic.
(2) Ii-bacteriostatic agents ezisebenza ngokukhawuleza ezifana ne-macrolides, i-tetracyclines kunye ne-amide alcohols ziphazamisa umphumo we-bactericidal wale mveliso kwaye akufanele zisetyenziswe kunye.
β- Lactam antibiotics. Isetyenziselwa ukunyanga usulelo lwebhaktiriya yegram-positive kunye nebhaktiriya yegram-negative enovelwano kwi-amoxicillin kwiinkukhu.
Kubalwa yile mveliso. Thatha ngomlomo: 0.2 ~ 0.3g yenkukhu nge-1kg ubunzima bomzimba. Amaxesha ama-2 ngosuku ngeentsuku ezi-5 ezilandelelanayo: isiselo esixutywe: inkukhu ye-0.6g nge-1L yamanzi kwi-3 ukuya kwiintsuku ezi-5 ezilandelelanayo.
Unempembelelo enamandla yokuphazamiseka kwizityalo eziqhelekileyo zesisu sesisu.
(1) Iinkukhu ezizalela amaqanda ukuze zityiwe ngabantu aziyi kusetyenziswa ngexesha lokubeka.
(2) Iintsholongwane ezikwigram-positive ezikwaziyo ukumelana nepenicillin akufuneki zisetyenziswe.
(3) Ukulungele ukusetyenziswa.
Idilesi:No.2 Xingding Road, Dingzhou City, Shijiazhuang, Hebei China
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