Amoxicillin Soluble Hmoov
Amoxicillin
Cov khoom no yog dawb los yog yuav luag dawb hmoov.
Pharmacodynamics Amoxicillin yog cov tshuaj tua kab mob B-lactam nrog cov kab mob dav dav. Cov tshuaj tua kab mob thiab kev ua haujlwm yog qhov tseem ceeb tib yam li ampicillin. Cov tshuaj tua kab mob tiv thaiv feem ntau cov kab mob gram-zoo yog me ntsis qis dua penicillin, thiab nws rhiab heev rau penicillinase, yog li nws tsis muaj txiaj ntsig tiv thaiv penicillin resistant Staphylococcus aureus. Nws muaj cov txiaj ntsig zoo ntawm cov kab mob gram-tsis zoo xws li Escherichia coli, Proteus, Salmonella, Haemophilus, Brucella thiab Pasteurella, tab sis cov kab mob no nquag ua rau cov tshuaj tiv thaiv. Nws tsis nkag siab rau Pseudomonas aeruginosa. Vim tias nws qhov nqus tau zoo hauv cov tsiaj txhu monogastric zoo dua li ampicillin, thiab nws cov ntshav concentration siab dua, nws muaj txiaj ntsig zoo rau kev kis kab mob. Nws muaj feem xyuam rau cov kab mob ua pa, tso zis, kab mob ntawm daim tawv nqaij thiab cov nqaij mos uas tshwm sim los ntawm cov kab mob rhiab heev.
Pharmacokinetics: amoxicillin yog qhov ruaj khov rau gastric acid, uas tau nqus los ntawm 74% ~ 92% tom qab kev tswj hwm qhov ncauj hauv cov tsiaj txhu. Cov ntsiab lus ntawm lub plab zom mov cuam tshuam rau tus nqi nqus, tab sis tsis cuam tshuam rau qib kev nqus, yog li kev sib xyaw pub mis siv tau. Tom qab kev tswj hwm qhov ncauj ntawm tib koob tshuaj, cov ntshav cov ntshav ntawm amoxicillin yog 1.5 ~ 3 npaug siab dua li ntawm ampicillin.
(1) Kev sib xyaw ua ke ntawm cov khoom no thiab aminoglycosides tuaj yeem ua rau muaj kev sib xyaw ua ke ntawm cov kab mob tom kawg, uas qhia txog kev sib koom ua ke.
(2) Cov kab mob bacteriostatic sai sai xws li macrolides, tetracyclines thiab amide alcohols cuam tshuam cov kab mob bactericidal ntawm cov khoom no thiab yuav tsum tsis txhob siv ua ke.
β-Lactam tshuaj tua kab mob. Nws yog siv los kho cov kab mob gram-positive thiab kab mob gram-negative rhiab rau amoxicillin hauv qaib.
Muab xam los ntawm cov khoom no. Noj qhov ncauj: 0.2 ~ 0.3g nqaij qaib ib 1kg lub cev hnyav. 2 zaug hauv ib hnub rau 5 hnub sib law liag: sib xyaw dej: 0.6g nqaij qaib ib 1L dej rau 3 mus rau 5 hnub sib law liag.
Nws muaj kev cuam tshuam muaj zog ntawm cov nroj tsuag ntawm lub plab zom mov.
(1) Cov qaib tso qe rau tib neeg noj yuav tsum tsis txhob siv thaum lub sij hawm tso.
(2) Cov kab mob Gram zoo resistant rau penicillin yuav tsum tsis txhob siv.
(3) Npaj siv.
Chaw nyob: No.2 Xingding Road, Dingzhou City, Shijiazhuang, Hebei Tuam Tshoj
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