Neomycin sulfate soluble ntụ ntụ
Neomycin sulfate
Ngwaahịa a bụ ụdị ọcha na ntụ ntụ edo edo.
Pharmacodynamics Neomycin bụ ọgwụ na-egbu egbu nke sitere na osikapa hydrogen glycoside. Ụdị nje bacteria ya yiri nke kanamycin. Ọ nwere mmetụta antibacterial siri ike na ọtụtụ nje bacteria gram-adịghị mma, dị ka Escherichia coli, Proteus, Salmonella na Pasteurella multocida, ma na-enwe mmetụta nke Staphylococcus aureus. Pseudomonas aeruginosa, gram-positive bacteria (ma e wezụga Staphylococcus aureus), Rickettsia, anaerobes na fungi na-eguzogide ọgwụ a.
Pharmacokinetics Neomycin anaghị adịkarị mgbe nchịkwa ọnụ na ngwa mpaghara gasịrị. Mgbe nchịkwa ọnụ gasịrị, naanị 3% nke ngụkọta neomycin na-apụ na mmamịrị, ọtụtụ n'ime ya na-esikwa na nsị na-enweghị mgbanwe. Ọrịa mucosa nke eriri afọ ma ọ bụ ọnya nwere ike ịbawanye nnabata. A na-etinye ọgwụ ahụ ngwa ngwa mgbe ịgba ọgwụ mgbochi ahụ gasịrị, usoro ime ya dịkwa ka nke kanamycin.
(1) Ejikọtara ya na ọgwụ nje macrolide, ọ nwere ike ịgwọ mastitis nke nje bacteria gram-positive kpatara.
(2) nchịkwa ọnụ nwere ike imetụta absorption nke digitalis, vitamin A ma ọ bụ vitamin B12.
(3) Ọ nwere mmetụta synergistic na penicillin ma ọ bụ cephalosporin.
(4) A na-eme ka mmetụta antibacterial nke ngwaahịa a dịkwuo mma na mpaghara alkaline, yana ọ dakọtara na ọgwụ alkaline (dị ka sodium bicarbonate, aminophylline na ndị ọzọ) nwere ike ịkwalite mmetụta antibacterial, mana nsi na-emekwa ka ọ dịkwuo mma. Antibacterial mgbe pH gafere 8.4 Kama nke ahụ, mmetụta ahụ na-ebelata.
(5) Cations dị ka Ca2+, Mg2+, Na+, NH na K+ nwere ike igbochi ọrụ antibacterial nke ngwaahịa ahụ.
(6) Ejikọtara ya na cephalosporin, dextran, diuretics dị ike (dị ka furosemide), erythromycin, wdg, ọ nwere ike ịkwalite ototoxicity nke ngwaahịa a.
(7) Skeletal muscle relaxants (dị ka succinylcholine chloride) ma ọ bụ ọgwụ nwere mmetụta a nwere ike iwusi Neuromuscular mgbochi mmetụta.
Ọgwụ nje aminoglycoside. A na-ejikarị ya akpọọ nkụ ọgwụgwọ ọrịa eriri afọ nke nje bacteria gram-adịghị mma kpatara.
Ngwaahịa a gbakọrọ ya. Ihe ọṅụṅụ agwakọta: 1.54 ~ 2.31g anụ ọkụkọ kwa 1L mmiri. Enwere ike iji ya mgbe niile maka ụbọchị 3-5.
Neomycin bụ ihe kacha egbu egbu na aminoglycosides, mana mmeghachi omume nsi ole na ole na-eme mgbe a na-enye ya ọnụ ma ọ bụ na mpaghara.
A gaghị eji ọkụkọ na-akụ akwa maka oriri mmadụ n'oge ịtọgbọrọ.
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