Neomycin Sulfate Soluble Powder
Neomycin sulfate
O lenei oloa o se ituaiga paʻepaʻe i le paʻu samasama malamalama.
Pharmacodynamics Neomycin ose vailaau antibacterial e maua mai le hydrogen glycoside araisa. O lona alaleo antibacterial e tutusa ma le kanamycin. E malosi lona aafiaga antibacterial i le tele o siama gram-negative, e pei ole Escherichia coli, Proteus, Salmonella ma Pasteurella multocida, ma e maaleale foi i Staphylococcus aureus. Pseudomonas aeruginosa, siama kalama (sei vagana ai Staphylococcus aureus), Rickettsia, anaerobes ma sigi e tetee i lenei oloa.
Pharmacokinetics Neomycin e seasea mitiia pe a uma le tuʻu gutu ma le faʻaoga i le lotoifale. A maeʻa le tuʻuina atu o le gutu, e naʻo le 3% o le aofaʻi o le neomycin e faʻamalo mai le urine, ma o le tele o mea e alu ese mai feces e aunoa ma se suiga. O le mumū o le mucosa o le intestinal poʻo le papala e mafai ona faʻateleina le faʻafefe. O le vailaʻau e vave faʻafefe pe a uma le tui, ma o lona gaioiga i totonu e tutusa ma le kanamycin.
(1) Faʻatasi ma vailaʻau faʻamaʻi macrolide, e mafai ona togafitia le mastitis e mafua mai i siama kalama.
(2) O le tu'u gutu e mafai ona a'afia ai le mitiia o numera, vaitamini A po'o vaitamini B12.
(3) E iai sona aafiaga fa'atasi ma le penicillin po'o le cephalosporin.
(4) O le aafiaga antibacterial o lenei oloa ua faaleleia i le siosiomaga alkaline, ma e fetaui ma vailaau alkaline (e pei o le sodium bicarbonate, aminophylline ma isi) e mafai ona faaleleia le aafiaga antibacterial, ae o le toxicity e tutusa foi le faaleleia. Antibacterial pe a sili atu le pH i le 8.4 I se isi itu, o le aʻafiaga e faʻavaivaia.
(5) Cations e pei o Ca2 +, Mg2 +, Na +, NH ma K + e mafai ona taofia le gaioiga antibacterial o le oloa.
(6) Faʻatasi ma cephalosporin, dextran, diuretics mamana (e pei o furosemide), erythromycin, ma isi, e mafai ona faʻaleleia le ototoxicity o lenei oloa.
(7) O mea faʻamalo maso o le skeletal (e pei o le succinylcholine chloride) poʻo vailaʻau faʻatasi ma lenei aʻafiaga e mafai ona faʻamalosia ai le Neuromuscular block effect.
Aminoglycoside antibiotic. E masani ona faʻaaogaina e faʻamago ai togafitiga faʻamaʻi gastrointestinal e mafua mai siama maʻaleʻale kalama-negative.
Fa'atatau e lenei oloa. Meainu fefiloi: 1.54~2.31g moa i le 1L vai. E mafai ona faʻaaogaina faʻaauau mo le 3 ~ 5 aso.
O le neomycin e sili ona oona i aminoglycosides, ae e itiiti ni mea oona e tupu pe a tuʻuina atu ile gutu poʻo le lotoifale.
O moa e tu'u fuamoa mo le taumafaina e le tagata e le tatau ona fa'aaogaina i le taimi e fa'ataoto ai.
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