Neomycin Sulfate Soluble Powder
Neomycin sulfate
Ichi chigadzirwa imhando yehupfu hweyero.
Pharmacodynamics Neomycin mushonga unorwisa mabhakitiriya unobva kuhydrogen glycoside mupunga. Iro antibacterial spectrum yakafanana neiyo kanamycin. Iyo ine yakasimba antibacterial mhedzisiro pane akawanda gram-negative mabhakitiriya, akadai seEscherichia coli, Proteus, Salmonella uye Pasteurella multocida, uye zvakare inonzwa kune Staphylococcus aureus. Pseudomonas aeruginosa, gram-positive bacteria (kunze kweStaphylococcus aureus), Rickettsia, anaerobes uye fungi inopikisa chigadzirwa ichi.
Pharmacokinetics Neomycin haiwanzo kutorwa mushure mekutonga nemuromo uye kushandiswa kwenzvimbo. Mushure mekutonga nemuromo, 3% chete yehuwandu hwehuwandu hweneomycin inobudiswa kubva muweti, uye yakawanda yacho inobudiswa kubva mumarara pasina kuchinja. Intestinal mucosa kuzvimba kana maronda anogona kuwedzera kubatwa. Mushonga unotorwa nekukurumidza mushure mejekiseni, uye maitiro ayo emukati akafanana neaya kanamycin.
(1) Yakasanganiswa ne macrolide antibiotics, inogona kurapa mastitis inokonzerwa ne gram-positive bacteria.
(2) Kudzora nemuromo kunogona kukanganisa kutorwa kwedigitalis, vhitamini A kana vhitamini B12.
(3) Iine synergistic effect ne penicillin kana cephalosporin.
(4) Iyo antibacterial mhedzisiro yechigadzirwa ichi inokwidziridzwa munharaunda yealkaline, uye inoenderana nealkaline zvinodhaka (senge sodium bicarbonate, aminophylline Uye zvichingodaro) inogona kuwedzera iyo antibacterial mhedzisiro, asi huturu hunowedzerwawo saizvozvo. Antibacterial apo pH inodarika 8.4 Pane zvinopesana, mhedzisiro yacho haina simba.
(5) Cations yakadai seCa2 +, Mg2 +, Na +, NH uye K + inogona kuvharidzira basa reantibacterial rechigadzirwa.
(6) Yakasanganiswa necephalosporin, dextran, ine simba diuretics (yakadai sefurosemide), erythromycin, nezvimwewo, inogona Kuwedzera ototoxicity yechigadzirwa ichi.
(7) Skeletal muscle relaxants (zvakadai se succinylcholine chloride) kana zvinodhaka zvine izvi zvinogona kusimbisa Neuromuscular block effect.
Aminoglycoside antibiotics. Inonyanya kushandiswa kuomesa kurapa gastrointestinal chirwere chinokonzerwa neanonzwa giremu-negative mabhakitiriya.
Yakaverengerwa nechigadzirwa ichi. Kunwa kwakasanganiswa: 1.54 ~ 2.31g huku pa1L yemvura. Inogona kushandiswa nguva dzose kwemazuva 3-5.
Neomycin ndiyo inonyanya kuchetura muaminoglycosides, asi mashoma ekuita muchetura anoitika kana ichiitwa nemuromo kana munharaunda.
Huku dzinokandira mazai kuti dzidyiwe nevanhu hadzifanirwe kushandiswa panguva yekukandira.
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