I-Neomycin Sulfate Powder encibilikayo
I-Neomycin sulfate
Lo mkhiqizo uwuhlobo lwempushana emhlophe kuya kokuphuzi.
I-Pharmacodynamics I-Neomycin iyisidakamizwa esilwa namagciwane esitholakala erayisini le-hydrogen glycoside. I-spectrum yayo ye-antibacterial ifana ne-kanamycin. Inomphumela onamandla we-antibacterial kuma-bacterium amaningi angenayo igram, njenge-Escherichia coli, i-Proteus, i-Salmonella ne-Pasteurella multocida, futhi iyazwela ku-Staphylococcus aureus. I-Pseudomonas aeruginosa, amagciwane e-gram-positive (ngaphandle kwe-Staphylococcus aureus), i-Rickettsia, i-anaerobes kanye nesikhunta amelana nalo mkhiqizo.
I-Pharmacokinetics I-Neomycin ayivami ukumuncwa ngemuva kokuphathwa ngomlomo kanye nokusetshenziswa kwendawo. Ngemuva kokuphathwa ngomlomo, kuphela u-3% yenani eliphelele le-neomycin elikhishwa emchamweni, futhi iningi lawo likhishwa endle ngaphandle kokushintsha. Ukuvuvukala kwe-mucosa emathunjini noma izilonda kungandisa ukumuncwa. Umuthi udonswa ngokushesha ngemva kokujova, futhi inqubo yawo yangaphakathi ifana neye-kanamycin.
(1) Ihlanganiswe nama-macrolide antibiotics, ingakwazi ukwelapha i-mastitis ebangelwa amagciwane egram-positive.
(2) Ukuphatha ngomlomo kungathinta ukumuncwa kwe-digitalis, uvithamini A noma uvithamini B12.
(3) Inomphumela we-synergistic nge-penicillin noma i-cephalosporin.
(4) Umphumela we-antibacterial walo mkhiqizo uthuthukiswa endaweni ye-alkaline, futhi uhambisana nezidakamizwa ze-alkaline (njenge-sodium bicarbonate, i-aminophylline nokunye) kungathuthukisa umphumela we-antibacterial, kodwa ubuthi bubuye buthuthukiswe ngokufanayo. I-antibacterial lapho i-pH idlula i-8.4 Ngokuphambene nalokho, umphumela uba buthaka.
(5) Ama-cations afana ne-Ca2+, Mg2+, Na+, NH kanye ne-K+ angavimbela umsebenzi we-antibacterial womkhiqizo.
(6) Ihlanganiswe ne-cephalosporin, i-dextran, i-diuretics enamandla (njenge-furosemide), i-erythromycin, njll., ingathuthukisa i-ototoxicity yalo mkhiqizo.
(7) Ukuphumula kwemisipha ye-skeletal (njenge-succinylcholine chloride) noma izidakamizwa ezinomphumela zingaqinisa umphumela we-Neuromuscular block.
Ama-antibiotic e-aminoglycoside. Ngokuyinhloko isetshenziselwa ukomisa ukwelapha izifo zamathumbu ezibangelwa amagciwane azwelayo egram-negative.
Kubalwe yilo mkhiqizo. Ukuphuza okuxubile: 1.54 ~ 2.31g yenkukhu nge-1L yamanzi. Ingasetshenziswa ngokuqhubekayo izinsuku ezingu-3-5.
I-Neomycin iwubuthi kakhulu kuma-aminoglycosides, kodwa kumbalwa ukusabela okunobuthi okwenzekayo lapho isetshenziswa ngomlomo noma endaweni.
Izinkukhu ezizalela amaqanda ukuze zidliwe abantu akufanele zisetshenziswe ngesikhathi sokubekela.
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