Erythromycin Thiocyanate Soluble Powder
Erythromycin
Ọja yi jẹ funfun tabi fere funfun lulú.
Pharmacodynamics Erythromycin jẹ egboogi macrolide. Ipa ọja yii lori awọn kokoro arun to dara giramu jẹ iru si penicillin, ṣugbọn irisi antibacterial rẹ gbooro ju pẹnisilini lọ. Awọn kokoro arun gram-positive ni Staphylococcus aureus (pẹlu Staphylococcus aureus penicillin sooro), pneumococcus, streptococcus, anthrax, erysipelas suis, listeria, clostridium putrescens, clostridium anthracis, ati bẹbẹ lọ , bbl Ni afikun, o tun ni ipa ti o dara lori Campylobacter, Mycoplasma, Chlamydia, Rickettsia ati Leptospira. Iṣẹ ṣiṣe antibacterial ti erythromycin thiocyanate ni ojutu ipilẹ jẹ imudara. Nigbati pH ba pọ si lati 5.5 si 8.5, iṣẹ ṣiṣe antibacterial n pọ si ni diėdiė. Pharmacokinetics Erythromycin ipilẹ ati stearate rọrun lati jẹ ibajẹ nipasẹ acid inu nigba ti a mu ni ẹnu. Iru ati fọọmu iwọn lilo ti iyọ Erythromycin, acidity ti inu ikun ati ounjẹ ti o wa ninu ikun gbogbo ni ipa lori bioavailability rẹ. Nikan awọn igbaradi ti a bo inu inu le jẹ gbigba dara julọ. Lẹhin gbigba, o ti pin kaakiri ni ọpọlọpọ awọn iṣan ati awọn omi ara, ṣugbọn ṣọwọn wọ inu omi cerebrospinal. Oṣuwọn abuda amuaradagba pilasima jẹ. 73% ~ 81% Apa kekere ti erythromycin jẹ metabolized bi N-methyl erythromycin aiṣiṣẹ ninu ẹdọ, eyiti o jẹ itujade ni akọkọ ninu bile apẹrẹ. Nikan 2% ~ 5% ti iwọn lilo ni a yọ jade ninu ito apẹrẹ.
(1) Ọja yii ko dara fun lilo ni akoko kanna bi awọn macrolides miiran ati awọn lincomamines nitori ibi-afẹde kanna.
(2) Nigbati o ba ni idapo pẹlu B-lactam, o ni ipa atagonistic.
(3) O le ṣe idiwọ eto oxidase cytochrome, ati pe o le ṣe idiwọ iṣelọpọ rẹ nigba lilo pẹlu awọn oogun kan.
Awọn egboogi macrolide. O ti wa ni lo lati toju àkóràn arun to šẹlẹ nipasẹ giramu-rere kokoro arun ati mycoplasma ni adie. Bi arun staphylococcal, streptococcal arun, onibaje atẹgun arun ati àkóràn rhinitis ni adie.
Ti ṣe iṣiro nipasẹ ọja yii. Ohun mimu ti a dapọ: 2.5g adie fun omi 1L. O le ṣee lo nigbagbogbo fun awọn ọjọ 3-5.
Lẹhin iṣakoso ẹnu, awọn ẹranko nigbagbogbo ni iwọn lilo ti o gbẹkẹle awọn rudurudu ifun, gẹgẹbi igbuuru.
(1) Adie ti o nfi ẹyin fun eniyan jẹ ko ṣee lo ni akoko gbigbe.
(2) Ọja yii ko yẹ ki o ni ibamu pẹlu awọn nkan ekikan.
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