Erythromycin Thiocyanate Ifu Yumuti
Erythromycin
Ibicuruzwa byera cyangwa ifu yera hafi.
Pharmacodynamics Erythromycin ni antibiyotike ya macrolide. Ingaruka yiki gicuruzwa kuri bagiteri-nziza ya bagiteri isa na penisiline, ariko spiba ya antibacterial ni nini kuruta penisiline. Indwara nziza ya bagiteri zirimo Staphylococcus aureus (harimo na penisiline irwanya Staphylococcus aureus), pneumococcus, streptococcus, anthrax, suis ya erysipelas, listeria, clostridium putrescens, clostridium anthracis, na bacteri za Sensitive gramm , n'ibindi, Byongeye kandi, bigira n'ingaruka nziza kuri Campylobacter, Mycoplasma, Chlamydia, Rickettsia na Leptospira. Igikorwa cya antibacterial ya erythromycin thiocyanate mumuti wa alkaline cyongerewe imbaraga. Iyo pH yiyongereye kuva 5.5 igera kuri 8.5, ibikorwa bya antibacterial byiyongera buhoro buhoro. Pharmacokinetics Erythromycin base na stearate biroroshye guteshwa agaciro na aside gastricike iyo ifashwe mukanwa. Ubwoko na dosiye y'umunyu wa Erythromycine, acide ya gastrointestinal tract hamwe nibiryo byo mu gifu byose bigira ingaruka kuri bioavailability. Gusa imyiteguro ya enteric yateguwe irashobora kwinjizwa neza. Nyuma yo kwinjizwa, ikwirakwizwa cyane mubice bitandukanye no mumazi yumubiri, ariko gake yinjira mumazi ya cerebrospinal. Igipimo cya plasma protein ihuza ni. 73% ~ 81% part Igice gito cya erythromycine gihindagurika nka N-methyl erythromycine idakora mu mwijima, ikaba isohoka cyane muri prototype. 2% ~ 5% gusa ya dose isohoka muminkari ya prototype.
(1) Iki gicuruzwa ntigikwiye gukoreshwa mugihe kimwe nizindi macrolide na lincomamine kubera intego imwe.
(2) Iyo ihujwe na B-lactam, igira ingaruka zo kurwanya.
(3) Irashobora guhagarika sisitemu ya okiside ya cytochrome, kandi irashobora guhagarika metabolisme yayo iyo ikoreshejwe nibiyobyabwenge.
Antibiyotike ya Macrolide. Ikoreshwa mu kuvura indwara zandura ziterwa na bagiteri-nziza ya bagiteri na mycoplasma mu nkoko. Nkindwara ya staphylococcal, indwara ya streptococcale, indwara zubuhumekero zidakira hamwe na rhinite yanduye mu nkoko.
Kubarwa niki gicuruzwa. Ikinyobwa kivanze: 2.5g inkoko kumazi 1L. Irashobora gukoreshwa ubudahwema iminsi 3 ~ 5.
Nyuma yo gutangwa mu kanwa, inyamaswa akenshi zifite urugero rwindwara ziterwa na gastrointestinal, nka diyare.
(1) Inkoko zitera amagi kugirango abantu barye ntizishobora gukoreshwa mugihe cyo gutera.
(2) Iki gicuruzwa ntigikwiye guhuzwa nibintu bya aside.
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