Erythromycin Thiocyanate Soluble Powder
Erythromycin
Ichi chigadzirwa chichena kana chinenge chena poda.
Pharmacodynamics Erythromycin ndeye macrolide antibiotic. Mhedzisiro yechigadzirwa ichi pa gram-positive bacteria yakafanana nepenicillin, asi antibacterial spectrum yayo yakakura kupfuura penicillin. Utachiona hwegiramu-positive hunosanganisira Staphylococcus aureus (kusanganisira penicillin inopikisa Staphylococcus aureus), pneumococcus, streptococcus, anthrax, erysipelas suis, listeria, clostridium putrescens, clostridium anthracis, nezvimwewo. Pasteurella, etc. Mukuwedzera, inewo migumisiro yakanaka paCampylobacter, Mycoplasma, Chlamydia, Rickettsia uye Leptospira. Iyo antibacterial chiitiko che erythromycin thiocyanate mune alkaline mhinduro yakasimbiswa. Kana iyo pH yakawedzera kubva pa5.5 kusvika ku8.5, iyo antibacterial chiitiko chakawedzera zvishoma nezvishoma. Pharmacokinetics Erythromycin base uye stearate zviri nyore kuderedzwa negastric acid kana inotorwa nemuromo. Mhando uye dosage fomu yeErythromycin munyu, acidity yemudumbu uye chikafu chiri mudumbu zvese zvinokanganisa bioavailability yayo. Chete enteric coated gadziriro inogona kubatwa zviri nani. Mushure mekutora, inoparadzirwa zvakanyanya mumhando dzakasiyana-siyana uye mvura yemuviri, asi kashoma inopinda mu cerebrospinal fluid. Iyo plasma protein inosunga mwero ndeye. 73% ~ 81% . Chikamu chidiki che erythromycin chinogadziriswa seN-methyl erythromycin isingashande muchiropa, iyo inonyanya kubudiswa mu prototype bile. Chete 2% ~ 5% yedosi inoburitswa mune prototype weti.
(1) Ichi chigadzirwa hachina kukodzera kushandiswa panguva imwe chete nemamwe macrolides uye lincomamines nekuda kwechinangwa chimwe chete.
(2) Kana yasanganiswa neB-lactam, ine antagonistic effect.
(3) Inogona kuvharidzira cytochrome oxidase system, uye inogona kuvharidzira metabolism yayo kana ichishandiswa nemimwe mishonga.
Macrolide antibiotics. Inoshandiswa kurapa zvirwere zvinotapukira zvinokonzerwa ne gram-positive bacteria uye mycoplasma muhuku. Zvakadai sechirwere che staphylococcal, chirwere che streptococcal, chirwere chisingaperi chekufema uye infectious rhinitis muhuku.
Yakaverengerwa nechigadzirwa ichi. Chinwiwa chakasanganiswa: 2.5g huku pa1 litre yemvura. Inogona kushandiswa nguva dzose kwemazuva 3-5.
Mushure mekutonga nemuromo, mhuka dzinowanzova nedosi inotsamira gastrointestinal kusagadzikana, senge manyoka.
(1) Huku dzinokandira mazai kuti dzidyiwe nevanhu hadzifanirwe kushandiswa panguva yekukandira.
(2) Ichi chigadzirwa hachifanirwe kuenderana nezvinhu zvine acidic.
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