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Levamisole 1000mg Bolus

Pharmacokinetics:Levamisole inotorwa kubva muura mushure memuromo uye kuburikidza neganda mushure mekushandiswa kwedermal, kunyange zvazvo bioavailabilities ichisiyana. Zvinonzi inogoverwa muviri wose. Levamisole inonyanya kushandiswa nemetabolized isingasviki 6% yakabudiswa isina kuchinjwa muweti. Plasma kubviswa kwehafu yeupenyu kwakatemwa kune akati wandei veterinary marudzi: Mombe 4-6 maawa; Imbwa 1.8-4 maawa; uye Swine 3.5-6.8 maawa. Metabolites inobudiswa muweti (kunyanya) uye tsvina.



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Pharmacokinetics

Levamisole inotorwa kubva muura mushure memuromo uye kuburikidza neganda mushure mekushandiswa kwedermal, kunyange zvazvo bioavailabilities ichisiyana. Zvinonzi inogoverwa muviri wose. Levamisole inonyanya kushandiswa nemetabolized isingasviki 6% yakabudiswa isina kuchinjwa muweti. Plasma kubviswa kwehafu yeupenyu kwakatemwa kune akati wandei veterinary marudzi: Mombe 4-6 maawa; Imbwa 1.8-4 maawa; uye Swine 3.5-6.8 maawa. Metabolites inobudiswa muweti (kunyanya) uye tsvina.

 

Zviratidzo

Levamisole inoratidzwa mukurapa nematodes akawanda mumombe, hwai nembudzi, nguruve, huku. Mumakwai nemombe, levamisole ine basa rakati nakei pakurwisa abomasal nematodes, nematodes emudumbu madiki (asina kunyanya kunyanyonakira Strongyloides spp.), matumbu mahombe (kwete Trichuris spp.), nemakonye emapapu. Mhando dzemhando dzemhando dzemhando dzemhando dzinowanzovharwa ne levamisole, dzinosanganisira: Haemonchus spp., Trichostrongylus spp., Osteragia spp., Cooperia spp., Nematodirus spp., Bunostomum spp., Oesophagostomum spp., Chabertia spp., uye Dictyopuulus. Levamisole hainyanyi kushanda kurwisa zvipembenene izvi zvisati zvakura uye kazhinji haishande mumombe (asi kwete hwai) pamhando dzemakonye akasungwa.

Munguruve, levamisole inoratidzwa pakurapa kweAscaris suum, Oesophagostomum spp., Strongyloides, Stephanurus, uye Metastrongylus.

Levamisole yakashandiswa mumbwa semicrofilaricide kurapa Dirofilaria immitis infection.

 

Contraindications/Kungwarira

Levamisole inopikiswa mumhuka dzinoyamwisa. Inofanirwa kushandiswa nekuchenjerera, kana zvachose, mumhuka dzakaremara zvakanyanya, kana dzine renal kana hepatic impairment. Shandisai nekuchenjerera kana, zvichida, kunonoka kushandiswa mumombe dzinenge dzakamanikidzwa nekuda kwejekiseni, kubvisa nyanga kana kukanda.

Iko hakuna ruzivo maererano nekuchengetedzwa kwechirwere ichi mumhuka dzine pamuviri. Kunyange zvazvo levamisole ichionekwa seyakachengetedzeka kuti ishandiswe mumhuka huru dzine mimba, shandisa chete kana mabhenefiti angangopfuura njodzi.

 

Zvakaipa Migumisiro/Yambiro

Migumisiro yakaipa iyo inogona kuonekwa mumombe inogona kusanganisira muromo-kupupuma kana hypersalivation, kufara kana kudedera, muromo wemuromo uye kudzungudza musoro. Migumisiro iyi inowanzoonekwa nepamusoro kudarika inokurudzirwa doses kana kana levamisole inoshandiswa panguva imwechete ne organophosphates. Zviratidzo zvinowanzopera mukati memaawa maviri. Pakuisa jekiseni mumombe, kuzvimba kunogona kuitika panzvimbo yejekiseni. Izvi zvinowanzopera mukati memazuva 7-14, asi zvinogona kunge zvisingabvumike mumhuka dzave pedyo nekuurayiwa.

 Mumakwai, levamisole inogona kukonzera kufara kwenguva pfupi mune dzimwe mhuka mushure mekutora. Mumbudzi, levamisole inogona kukonzera kuora mwoyo, hyperesthesia uye salivation.
 Munguruve, levamisole inogona kukonzera mate kana muromo kupupuma furo. Nguruve ine utachiona hwemapapu inogona kutanga kukosora kana kurutsa.

 Migumisiro yakaipa inogona kuonekwa muimbwa inosanganisira kuvhiringidzika kweGI (kazhinji kurutsa, manyoka), neurotoxicity (kufema, kuzununguka, kusagadzikana kana mamwe maitiro ekuchinja), agranulocytosis, dyspnea, pulmonary edema, immune-mediated skin eruptions (erythroedema, erythema multiforme, chepfu. epidermal necrolysis) uye kuneta.

 Migumisiro yakaipa inoonekwa mumakati inosanganisira hypersalivation, kufara, mydriasis uye kurutsa.
 

Dosage uye Administration

Yekutonga nemuromo.

The general dosage is 5-7.5 mg Levamisole per kg bodyweight.

Kuti uwane rumwe ruzivo nezve bolus yega yega, ona tafura pazasi.

Bolus Dosage:

150mg 1 bolus pa25kg yehuremu hwemuviri.

600mg 1 bolus pa100kg yehuremu hwemuviri.

1000mg 1 bolus pa150kg yehuremu hwemuviri.

 

Withdrawal Period

Mombe (nyama & offal): 5 mazuva.

Hwai (nyama & offal): mazuva mashanu.

Haufanirwe kushandiswa mumhuka dzinogadzira mukaka uchidyiwa nevanhu.

 

Storage

Iyo yakanyanya kukurudzirwa tembiricha yekuchengetedza i30 ℃.

Yambiro:Gara kure nekusvikirwa nevana.

 

Kana iwe uchifarira zvigadzirwa zvedu, unogona kusarudza kusiya ruzivo rwako pano, uye isu tichabatana newe munguva pfupi.


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Kana iwe uchifarira zvigadzirwa zvedu, unogona kusarudza kusiya ruzivo rwako pano, uye isu tichabatana newe munguva pfupi.


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Kana iwe uchifarira zvigadzirwa zvedu, unogona kusarudza kusiya ruzivo rwako pano, uye isu tichabatana newe munguva pfupi.


Kana iwe uchifarira zvigadzirwa zvedu, unogona kusarudza kusiya ruzivo rwako pano, uye isu tichabatana newe munguva pfupi.