Enrofloxacin duritaan
Enrofloxacin
Alaabtani waa mid aan midab lahayn ama midab huruud ah oo caddaan ah.
Pharmacodynamic Enrofloxacin waa daawo bakteeriya-bakteeriya ah oo ballaaran oo si gaar ah loogu isticmaalo xayawaanka fluoroquinolone. Waayo e. coli, salmonella, klebsiella, brucella, pasteurella, pleuropneumonia actinobacillus, erysipelas, bacillus proteus, clayey bakteeriyada Mr Charest, corynebacterium suppurative, bakteeriyada dhariga dhiiga ee jabtay, staphylococcus aureus, mycoplasma, chlamygin, iyo wixii la mid ah oo dhan waxay leeyihiin saameyn wanaagsan oo ah peruudose. iyo streptococcus waa daciif, saameyn daciif ah bakteeriyada anaerobic. Waxay leedahay saameyn cad ka dib-bakteeriyadu waxay ku leedahay bakteeriyada xasaasiga ah. Habka ficilka bakteeriyada ee alaabtani waa in la joojiyo wareegga DNA-da bakteeriyada, farageliya soo-celinta, qorista iyo hagaajinta dib-u-habaynta DNA-da bakteeriyada, bakteeriyadu si caadi ah uma kori karto oo uma taran karto oo dhimanayso.
Pharmacokinetics Daawadu si dhakhso ah oo buuxda ayaa loo nuugay cirbadeynta muruqa. bioavailability-ku wuxuu ahaa 91.9% doofaarka iyo 82% lo'da. Waxay si weyn ugu qaybsan tahay xayawaanka waxayna si fiican u geli kartaa unugyada iyo dareeraha jidhka. Marka laga reebo dareeraha cerebrospinal, fiirsashada daawada ee ku dhawaad dhammaan unugyada ayaa ka sarreeya tan plasma. Dheef-shiid kiimikaad ee ugu weyn waa ka saarida ethyl ee giraanta 7-piperazine si loo soo saaro ciprofloxacin, oo ay ku xigto oksaydheynta iyo glucuronic acid. Inta badan kelyaha (dheecaanka tubbada kelyaha iyo shaandhaynta glomerular), dheecaanka 15% ~ 50% oo ah qaabka asalka ah ee kaadida. Ciribtirka nolosha nuska ah ee cirbadeynta muruqyada gudaha waxay ahayd 5.9 saacadood lo'da caanaha, 1.5 ~ 4.5 saacadood oo idaha ah, iyo 4.6 saacadood oo doofaarro ah.
(1) Alaabtani waxay leedahay saameyn isku-dhafan marka lagu daro aminoglycosides ama penicillin-spectrum ballaaran.
(2) Ca2+, Mg2+, Fe3+, Al3+ iyo ayoonooyinka kale ee birta culus waxay ku dhayalsan karaan alaabtan, taasoo saamaynaysa nuugista.
(3) Marka lagu daro theophylline iyo kafeyn, heerka isku xirnaanta borotiinka balaasmaha waa la dhimaa, iyo diirada theophylline iyo kafeyn ee dhiiga si aan caadi aheyn ayaa u kordhay.
Xitaa waxay muuqdaan calaamadaha sunta theophylline.
(4) Alaabtani waxay leedahay saamaynta joojinta enzymes daroogada beerka, taas oo yarayn karta heerka nadiifinta ee daawooyinka inta badan metabolized beerka, iyo kordhinta diiradda dhiigga ee daroogada.
[Doorka iyo isticmaalka] Quinolones daawooyinka bakteeriyada. Waxaa loo isticmaalaa cudurrada bakteeriyada iyo caabuqyada mycoplasma ee xoolaha iyo digaagga.
Daawooyinka bakteeriyada ee Quinolones. Waxaa loo isticmaalaa cudurrada bakteeriyada iyo caabuqyada mycoplasma ee xoolaha iyo digaagga.
Duritaan muruqa ah: hal qiyaas, 0.025ml 1kg miisaanka jirka ee lo'da, idaha iyo doofaarka; Eyda, bisadaha, bakaylaha 0.025-0.05 ml. Isticmaal hal ama laba jeer maalintii laba ilaa saddex maalmood.
(1) Carjawda carjawda waxay ku dhacdaa xayawaanka da'da yar, oo saameeya horumarka lafaha oo keena claudication iyo xanuun.
(2) Dareen-celinta hab-dhiska dheefshiidka waxaa ka mid ah matag, cunto xumo, shuban, iwm.
(3) Dareen-celinta maqaarka waxaa ka mid ah erythema, cuncun, urtikaria iyo falcelinta sawir-qaadista.
(4) Dareen-celinta xasaasiyadda, ataxia iyo suuxdin ayaa marmar lagu arkaa eeyaha iyo bisadaha.
(1) Waxay ku yeelan kartaa saamaynta kicinta ee nidaamka dhexe waxayna keeni kartaa suuxdin. Waa in si taxadar leh loo isticmaalo eeyaha qaba suuxdin.
(2) Hilibka cuna iyo xayawaanka leh shaqada kelyaha oo liidata ayaa si taxadar leh loo isticmaalo, marmar bay kaadida soo kicin karaan.
(3) Alaabtani kuma habboona eeyaha ka hor 8 toddobaad jir.
(4) Noocyada u adkeysiga daawada ee alaabtan ayaa sii kordhaya, markaa waa in aan loo isticmaalin qiyaasta daweynta hoose muddo dheer.
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